Compile Data Set for Download or QSAR
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Found 17 Enz. Inhib. hit(s) with all data for entry = 50038877
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50124303(3-[16-carbamoyl-31-carbamoylmethyl-10-(2-carboxyet...)
Affinity DataIC50:  1.50E+4nMAssay Description:Binding affinity to GST-tagged recombinant Grb2 SH2 domain by Biacore assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50294422(4-{[(9S,15R,18S,21S)-15-carbamoyl-21-(carbamoylmet...)
Affinity DataKd:  880nMAssay Description:Binding affinity to GST-tagged recombinant Grb2 SH2 domain by Biacore assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50378056(CHEMBL1627249)
Affinity DataKd:  4.80E+3nMAssay Description:Binding affinity to GST-tagged recombinant Grb2 SH2 domain by Biacore assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50378057(CHEMBL1627267)
Affinity DataKd:  1.29E+3nMAssay Description:Binding affinity to GST-tagged recombinant Grb2 SH2 domain by Biacore assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50378057(CHEMBL1627267)
Affinity DataKd:  2.14E+3nMAssay Description:Binding affinity to GST-tagged recombinant Grb2 SH2 domain by Biacore assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50378058(CHEMBL1627247)
Affinity DataKd:  1.72E+3nMAssay Description:Binding affinity to GST-tagged recombinant Grb2 SH2 domain by Biacore assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50378058(CHEMBL1627247)
Affinity DataKd:  1.36E+3nMAssay Description:Binding affinity to GST-tagged recombinant Grb2 SH2 domain by Biacore assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50378059(CHEMBL1627251)
Affinity DataKd:  1.76E+3nMAssay Description:Binding affinity to GST-tagged recombinant Grb2 SH2 domain by Biacore assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50378059(CHEMBL1627251)
Affinity DataKd:  1.56E+3nMAssay Description:Binding affinity to GST-tagged recombinant Grb2 SH2 domain by Biacore assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50294415(4-{[(9S,15R,18S,21S)-15-carbamoyl-21-(carbamoylmet...)
Affinity DataKd:  2.71E+3nMAssay Description:Binding affinity to GST-tagged recombinant Grb2 SH2 domain by Biacore assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50294416(4-{[(9S,15R,18S,21S)-15-carbamoyl-21-(carbamoylmet...)
Affinity DataKd:  1.05E+3nMAssay Description:Binding affinity to GST-tagged recombinant Grb2 SH2 domain by Biacore assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50294417(4-{[(9S,15R,18S,21S)-15-carbamoyl-21-(carbamoylmet...)
Affinity DataKd:  1.06E+3nMAssay Description:Binding affinity to GST-tagged recombinant Grb2 SH2 domain by Biacore assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50294418(4-{[(9S,15R,18S,21S)-15-carbamoyl-21-(carbamoylmet...)
Affinity DataKd:  1.42E+3nMAssay Description:Binding affinity to GST-tagged recombinant Grb2 SH2 domain by Biacore assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50294419(3-[(5S,8S,11S,14S,17R)-17-carbamoyl-11-(carbamoylm...)
Affinity DataKd:  3.60E+3nMAssay Description:Binding affinity to GST-tagged recombinant Grb2 SH2 domain by Biacore assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50124303(3-[16-carbamoyl-31-carbamoylmethyl-10-(2-carboxyet...)
Affinity DataKd:  2.50E+4nMAssay Description:Binding affinity to GST-tagged recombinant Grb2 SH2 domain by Biacore assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50294420(4-[(9S,12S,19S,22S)-12-amino-22-(carbamoylmethyl)-...)
Affinity DataKd:  7.55E+3nMAssay Description:Binding affinity to GST-tagged recombinant Grb2 SH2 domain by Biacore assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50294421(4-{[(9S,15R,18S,21S)-15-carbamoyl-21-(carbamoylmet...)
Affinity DataKd:  359nMAssay Description:Binding affinity to GST-tagged recombinant Grb2 SH2 domain by Biacore assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed