Compile Data Set for Download or QSAR
maximum 50k data
Found 32 Enz. Inhib. hit(s) with all data for entry = 50033146
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50340362(2-(4-chloro-2-fluorophenyl)-1-{3-[4-(3-acetylamino...)
Affinity DataIC50:  1nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50340346(2-(4-chlorophenyl)-1-{3-[4-(3-acetylaminophenyl)pi...)
Affinity DataIC50:  1nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50340341(2-phenyl-1-{3-[4-(3-acetylaminophenyl)piperidin-1-...)
Affinity DataIC50:  2nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50340349(2-(4-trifluoromethylphenyl)-1-{3-[4-(3-acetylamino...)
Affinity DataIC50:  3nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50340360(2-(2,4-dichlorophenyl)-1-{3-[4-(3-acetylaminopheny...)
Affinity DataIC50:  3nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50340346(2-(4-chlorophenyl)-1-{3-[4-(3-acetylaminophenyl)pi...)
Affinity DataIC50:  3nMAssay Description:Inhibition hERG by patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50340364(2-(2-chloro-4-fluorophenyl)-1-{3-[4-(3-acetylamino...)
Affinity DataIC50:  4nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50340363(2-(3,4-difluorophenyl)-1-{3-[4-(3-acetylaminopheny...)
Affinity DataIC50:  4nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50340345(2-(3-chlorophenyl)-1-{3-[4-(3-acetylaminophenyl)pi...)
Affinity DataIC50:  5nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50340354(2-(4-bromophenyl)-1-{3-[4-(3-acetylaminophenyl)pip...)
Affinity DataIC50:  5nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50340367(2-(4-chlorophenyl)-1-{3-[4-(3-isobutyrylaminopheny...)
Affinity DataIC50:  5nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50340351(2-(3-methoxyphenyl)-1-{3-[4-(3-acetylaminophenyl)p...)
Affinity DataIC50:  7nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50340357(2-(4-biphenyl)-1-{3-[4-(3-acetylaminophenyl)piperi...)
Affinity DataIC50:  8nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50340352(2-(4-methoxyphenyl)-1-{3-[4-(3-acetylaminophenyl)p...)
Affinity DataIC50:  9nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50340344(2-(2-chlorophenyl)-1-{3-[4-(3-acetylaminophenyl)pi...)
Affinity DataIC50:  10nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50340359(2-(4-cyanophenyl)-1-{3-[4-(3-acetylaminophenyl)pip...)
Affinity DataIC50:  16nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50340368(2-(4-chlorophenyl)-1-{3-[4-(3-benzoylaminophenyl)p...)
Affinity DataIC50:  19nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50340361(2-(3,4-dichlorophenyl)-1-{3-[4-(3-acetylaminopheny...)
Affinity DataIC50:  24nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50340342(2-phenyl-1-{4-[4-(3-acetylaminophenyl)piperidin-1-...)
Affinity DataIC50:  29nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50340348(2-(3-trifluoromethylphenyl)-1-{3-[4-(3-acetylamino...)
Affinity DataIC50:  30nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50340355(2-(4-Ethylphenyl)-1-{3-[4-(3-acetylaminophenyl)pip...)
Affinity DataIC50:  32nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50340358(2-(4-phenoxyphenyl)-1-{3-[4-(3-acetylaminophenyl)p...)
Affinity DataIC50:  42nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50340347(2-(2-trifluoromethylphenyl)-1-{3-[4-(3-acetylamino...)
Affinity DataIC50:  50nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50340353(2-(4-Fluorophenyl)-1-{3-[4-(3-acetylaminophenyl)pi...)
Affinity DataIC50:  56nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50340356(2-(4-isopropylphenyl)-1-{3-[4-(3-acetylaminophenyl...)
Affinity DataIC50:  60nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50340343(2-phenyl-1-{5-[4-(3-acetylaminophenyl)piperidin-1-...)
Affinity DataIC50:  74nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50340370(2-(4-chlorophenyl)-1-{3-[4-(3-(4-methylbenzoylamin...)
Affinity DataIC50:  213nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50340369(2-(4-chlorophenyl)-1-{3-[4-(3-(3-chlorobenzoylamin...)
Affinity DataIC50:  300nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50340350(2-(2-methoxyphenyl)-1-{3-[4-(3-acetylaminophenyl)p...)
Affinity DataIC50:  747nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50340366(2-(4-chlorophenyl)-1-{5-[4-(4-acetylaminophenyl)pi...)
Affinity DataIC50:  5.38E+3nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50340365(2-(4-chlorophenyl)-1-{5-[4-(2-acetylaminophenyl)pi...)
Affinity DataIC50: >6.00E+3nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50340340(2-phenyl-1-{2-[4-(3-acetylaminophenyl)piperidin-1-...)
Affinity DataIC50:  1.00E+4nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed