Compile Data Set for Download or QSAR
maximum 50k data
Found 17 Enz. Inhib. hit(s) with all data for entry = 50039472
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350709(CHEMBL1812080)
Affinity DataIC50:  130nMAssay Description:Antagonist activity at Vibrio fischeri ESI 114 (delta-LuxI) LuxR assessed as inhibition of OdDHL-induced quorum sensing activation after 8 hrs by bet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350708(CHEMBL1814832)
Affinity DataIC50:  310nMAssay Description:Antagonist activity at Vibrio fischeri ESI 114 (delta-LuxI) LuxR assessed as inhibition of OdDHL-induced quorum sensing activation after 8 hrs by bet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350704(CHEMBL1814829)
Affinity DataIC50:  350nMAssay Description:Antagonist activity at Vibrio fischeri ESI 114 (delta-LuxI) LuxR assessed as inhibition of OdDHL-induced quorum sensing activation after 8 hrs by bet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350711(CHEMBL1812089)
Affinity DataIC50:  350nMAssay Description:Antagonist activity at Vibrio fischeri ESI 114 (delta-LuxI) LuxR assessed as inhibition of OdDHL-induced quorum sensing activation after 8 hrs by bet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350703(CHEMBL1814828)
Affinity DataIC50:  450nMAssay Description:Antagonist activity at Vibrio fischeri ESI 114 (delta-LuxI) LuxR assessed as inhibition of OdDHL-induced quorum sensing activation after 8 hrs by bet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350710(CHEMBL1812087)
Affinity DataIC50:  770nMAssay Description:Antagonist activity at Vibrio fischeri ESI 114 (delta-LuxI) LuxR assessed as inhibition of OdDHL-induced quorum sensing activation after 8 hrs by bet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350707(CHEMBL1814831)
Affinity DataIC50:  840nMAssay Description:Antagonist activity at Vibrio fischeri ESI 114 (delta-LuxI) LuxR assessed as inhibition of OdDHL-induced quorum sensing activation after 8 hrs by bet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein TraR(Rhizobium radiobacter)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350703(CHEMBL1814828)
Affinity DataIC50:  1.80E+3nMAssay Description:Antagonist activity at Agrobacterium tumefaciens WCF (pCF372) TraR assessed as inhibition of OdDHL-induced quorum sensing activation after 8 hrs by b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein TraR(Rhizobium radiobacter)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350706(CHEMBL1811922)
Affinity DataIC50:  2.80E+3nMAssay Description:Antagonist activity at Agrobacterium tumefaciens WCF (pCF372) TraR assessed as inhibition of OdDHL-induced quorum sensing activation after 8 hrs by b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein TraR(Rhizobium radiobacter)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350705(CHEMBL1814827)
Affinity DataIC50:  3.20E+3nMAssay Description:Antagonist activity at Agrobacterium tumefaciens WCF (pCF372) TraR assessed as inhibition of OdDHL-induced quorum sensing activation after 8 hrs by b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein TraR(Rhizobium radiobacter)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350708(CHEMBL1814832)
Affinity DataIC50:  1.00E+4nMAssay Description:Antagonist activity at Agrobacterium tumefaciens WCF (pCF372) TraR assessed as inhibition of OdDHL-induced quorum sensing activation after 8 hrs by b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350705(CHEMBL1814827)
Affinity DataIC50:  1.30E+4nMAssay Description:Antagonist activity at Pseudomonas aeruginosa PAO1 MW1 (pUM15) LasR assessed as inhibition of OdDHL-induced quorum sensing activation after 8 hrs by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350703(CHEMBL1814828)
Affinity DataEC50:  3.20E+3nMAssay Description:Agonist activity at Pseudomonas aeruginosa PAO1 MW1 (pUM15) LasR after 8 hrs by beta-galactosidase reporter gene assay relative to OdDHLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350706(CHEMBL1811922)
Affinity DataEC50:  2.10E+4nMAssay Description:Agonist activity at Pseudomonas aeruginosa PAO1 MW1 (pUM15) LasR after 8 hrs by beta-galactosidase reporter gene assay relative to OdDHLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350705(CHEMBL1814827)
Affinity DataEC50:  1.30E+4nMAssay Description:Agonist activity at Pseudomonas aeruginosa PAO1 MW1 (pUM15) LasR after 8 hrs by beta-galactosidase reporter gene assay relative to OdDHLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein TraR(Rhizobium radiobacter)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350704(CHEMBL1814829)
Affinity DataEC50:  2.00E+4nMAssay Description:Agonist activity at Agrobacterium tumefaciens WCF (pCF372) TraR after 8 hrs by beta-galactosidase reporter gene assay relative to OdDHLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350712(CHEMBL1812084)
Affinity DataEC50:  1.10E+4nMAssay Description:Agonist activity at Vibrio fischeri ESI 114 (delta-LuxI) LuxR after 8 hrs by beta-galactosidase reporter gene assay relative to OdDHLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed