Compile Data Set for Download or QSAR
maximum 50k data
Found 8 Enz. Inhib. hit(s) with all data for entry = 6067
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Sharpe & Dohme

US Patent
LigandPNGBDBM107106(US8592371, 7 | US9278976, (3S,5R)-5-[2-(cyclopropa...)
Affinity DataIC50:  1nMAssay Description:Enzyme assay using dipeptidyl peptidase-IV.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Sharpe & Dohme

US Patent
LigandPNGBDBM107103(US8592371, 5 | US9278976, (3S,5R)-5-[2-(cyclopenta...)
Affinity DataIC50:  1.30nMAssay Description:Enzyme assay using dipeptidyl peptidase-IV.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Sharpe & Dohme

US Patent
LigandPNGBDBM107102(US8592371, 4 | US9278976, (3S,5R)-5-[2-(cyclopenta...)
Affinity DataIC50:  1.60nMAssay Description:Enzyme assay using dipeptidyl peptidase-IV.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Sharpe & Dohme

US Patent
LigandPNGBDBM107104(US8592371, 6 | US9278976, (3S,5R)-5-[1-(cyclopropa...)
Affinity DataIC50:  1.60nMAssay Description:Enzyme assay using dipeptidyl peptidase-IV.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Sharpe & Dohme

US Patent
LigandPNGBDBM107105(US8592371, 8 | US9278976, (3S,5R)-5-[2-(cyclopropa...)
Affinity DataIC50:  1.90nMAssay Description:Enzyme assay using dipeptidyl peptidase-IV.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Sharpe & Dohme

US Patent
LigandPNGBDBM107100(US8592371, 2 | US9278976, (3S,5R)-5-{2-methanesulf...)
Affinity DataIC50:  2.20nMAssay Description:Enzyme assay using dipeptidyl peptidase-IV.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Sharpe & Dohme

US Patent
LigandPNGBDBM107099(US8592371, 1 | US9278976, (3S,5R)-2-(2,5-difluorop...)
Affinity DataIC50:  2.5nMAssay Description:Enzyme assay using dipeptidyl peptidase-IV.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Sharpe & Dohme

US Patent
LigandPNGBDBM107101(US8592371, 3)
Affinity DataIC50:  2.60nMAssay Description:Enzyme assay using dipeptidyl peptidase-IV.More data for this Ligand-Target Pair
In DepthDetails US Patent