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Target
Platelet-activating factor receptor
Ligand
BDBM50118195
Substrate
n/a
Meas. Tech.
ChEMBL_155144 (CHEMBL760185)
Ki
560.0±n/a nM
Citation
 Strømgaard, K; Saito, DR; Shindou, H; Ishii, S; Shimizu, T; Nakanishi, K Ginkgolide derivatives for photolabeling studies: preparation and pharmacological evaluation. J Med Chem 45:4038-46 (2002) [PubMed]  Article 
Target
Name:
Platelet-activating factor receptor
Synonyms:
PAF-R | PTAFR_MOUSE | Platelet activating factor receptor | Platelet-activating factor receptor | Ptafr
Type:
PROTEIN
Mol. Mass.:
39163.36
Organism:
Mus musculus
Description:
ChEMBL_155144
Residue:
341
Sequence:
MEHNGSFRVDSEFRYTLFPIVYSVIFILGVVANGYVLWVFANLYPSKKLNEIKIFMVNLTMADLLFLITLPLWIVYYYNEGDWILPNFLCNVAGCLFFINTYCSVAFLGVITYNRYQAVAYPIKTAQATTRKRGISLSLIIWVSIVATASYFLATDSTNLVPNKDGSGNITRCFEHYEPYSVPILVVHVFIAFCFFLVFFLIFYCNLVIIHTLLTQPMRQQRKAGVKRRALWMVCTVLAVFIICFVPHHVVQLPWTLAELGYQTNFHQAINDAHQITLCLLSTNCVLDPVIYCFLTKKFRKHLSEKFYSMRSSRKCSRATSDTCTEVIVPANQTPIVSLKN
  
Inhibitor
Name:
BDBM50118195
Synonyms:
3'-(tert-butyl)-4,9',14'-trihydroxy-2-methoxy-10'-methylspiro[tetrahydrofuran-3,2'-(6',12'-dioxatetracyclo[6.6.0.01,5.09,13]tetradecane)]-5,7',11'-trione | CHEMBL338808
Type:
Small organic molecule
Emp. Form.:
C21H28O10
Mol. Mass.:
440.441
SMILES:
COC1OC(=O)[C@H](O)C11[C@@H](CC2OC(=O)C3[C@@]4(O)[C@H](C)C(=O)O[C@H]4[C@H](O)[C@]123)C(C)(C)C
Structure:
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