Target Names are taken from UniProtKB. To view the associated UniProt page, click on the UniProt ID. When we have data for a given Target in multiple species or for mutants of a given Target, we provide a header row (upper case, bold font) with all of the data followed by a separate for each species or variant of the Target.
Target Name
Organism
Affinity Links
Articles
UniProts
Files
Human
IC50: 113
Human
Rapamycin-insensitive companion of mTOR/Serine/threonine-protein kinase mTOR/Target of rapamycin complex 2 subunit MAPKAP1/Target of rapamycin complex subunit LST8 P42345 Q6R327 Q9BPZ7 Q9BVC4
Human
IC50: 1
Human
Human
IC50: 233
Mitogen-activated protein kinase kinase kinase 7/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1 O43318 Q15750
Human
IC50: 196
Acinetobacter baumannii (AYE strain)
Acinetobacter baumannii (AYE strain)
Human
IC50: 11
Human
IC50: 11
Human herpesvirus 1 (strain SC16) (HHV-1) (Human herpes simplex virus1)
Varicella-zoster virus (strain Dumas) (HHV-3) (Human herpesvirus 3)
IC50: 55
Human herpesvirus 1 (strain SC16) (HHV-1) (Human herpes simplex virus1)
Human
EC50: 22
Rattus norvegicus
Human
IC50: 11
Mus musculus (Mouse)
Rattus norvegicus (Rat)
Human
IC50: 11
Human
Human
IC50: 1
Human
Rattus norvegicus
Mus musculus
IC50: 43
Mus musculus
EC50: 5
IC50: 2
Human
Rattus norvegicus (Rat)
Rattus norvegicus (rat)
Human
Cavia porcellus
IC50: 1
Mus musculus
Human
Rattus norvegicus
Human
Rattus norvegicus
Human
Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv)
Kd: 3
Haemophilus influenzae (strain ATCC 51907 / DSM 11121 / KW20 / Rd)
IC50: 31
Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22644 / CIP 104116 / JCM14847 / LMG 12228 / 1C / PRS 101 / PAO1)
Staphylococcus aureus (strain NCTC 8325 / PS 47)
Kd: 3
Bos taurus
Bos taurus
IC50: 4
Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv)
IC50: 12
Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv)
IC50: 6
Human
Human
IC50: 1
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform/Tyrosine-protein kinase ABL1 P00519 P42336
Human
IC50: 1
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform/Tyrosine-protein kinase ABL1 O00329 P00519
Human
IC50: 1
Human
IC50: 1
Human
IC50: 41
Human
Human
Human
IC50: 1
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform/Tyrosine-protein kinase HCK P08631 P42336
Human
IC50: 1
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform/Tyrosine-protein kinase HCK O00329 P08631
Human
IC50: 1
Human
IC50: 1
Human
IC50: 204
Mus musculus
IC50: 1
Non-receptor tyrosine-protein kinase TYK2/Tyrosine-protein kinase JAK1/Tyrosine-protein kinase JAK2 O60674 P23458 P29597
Human
IC50: 31
Non-receptor tyrosine-protein kinase TYK2/Tyrosine-protein kinase JAK1/Tyrosine-protein kinase JAK2 O60674 P23458 P29597
Human
IC50: 31
Non-receptor tyrosine-protein kinase TYK2/Tyrosine-protein kinase JAK1/Tyrosine-protein kinase JAK2/Tyrosine-protein kinase JAK3 O60674 P23458 P29597 P52333
Human
IC50: 79
Human
IC50: 74
Non-receptor tyrosine-protein kinase TYK2/Tyrosine-protein kinase JAK1/Tyrosine-protein kinase JAK2/Tyrosine-protein kinase JAK3 O60674 P23458 P29597 P52333
Human
IC50: 79
Human
IC50: 1
Tyrosine-protein kinase Mer
IC50: 76
Tyrosine-protein kinase transforming protein Src [144-247,E177Q,S178L,E179A,T180R,T181V,C186A,K201L] P63185
Rous sarcoma virus (Virus)
Kd: 2
Tyrosine-protein kinase transforming protein Src [144-247,E177R,S178L,E179Q,T180R,T181V,C186A,K201L] P63185
Rous sarcoma virus (Virus)
Kd: 2
Rous sarcoma virus (Virus)
Kd: 2
Rous sarcoma virus (Virus)
Kd: 2
Rattus norvegicus (rat)
Human
Human
Human
Human
Human
Human
Human
Human
Curated by BindingDB
Curated by ChEMBL