Search by Compound Name
Compounds Sorted by Binding Targets per Compound
1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 2930 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 50 51 52 53 54 55
56 57 58 59 60 61 62 63 64 65 66 67 68 69 70 73 74 75 76 77 79 81 84 86 89 95
96 100 108 109 120 124 130 137 143 154 156 168 186 224 240 259 276 278 284 303
304 310 315 323 339 369 370 371 372 373 374 375 376 377 378 380 381 383 384
385 386 388 389 390 391 392 393 394 395 397 398 401 403 404 406 408 418 427
429 443 447 515
Compounds Sorted Alphabetically
Compound Name (alphabetical)
Binding Targets
Enz. Inhib. Data
ITC Data
Alternate Compound Names
- β-Carbonic anhydrase 2 (CA 2)
- 5-HT3A Serotonin Receptor
- 5-hydroxytryptamine receptor 1A
- 5-hydroxytryptamine receptor 2A
- Alpha carbonic anhydrase
- Alpha-1A adrenergic receptor
- Astrosclerin-3
- Beta-2 adrenergic receptor
- Beta-carbonic anhydrase
- Bile salt export pump
- Bile salt export pump (BSEP)
- Carbonate dehydratase
- Carbonic Anhydrase III
- Carbonic Anhydrase IV
- Carbonic anhydrase
- Carbonic anhydrase 1
- Carbonic anhydrase 12
- Carbonic anhydrase 2
- Carbonic anhydrase 6 (CA-VI)
- Carbonic anhydrase 9
- Carbonic anhydrase, alpha family
- Carbonic anhydrases; II & IX
- Cytochrome P450 2J2
- D(1A) dopamine receptor
- D(1B) dopamine receptor
- D(2) dopamine receptor
- D(3) dopamine receptor
- D(4) dopamine receptor
- DRD1
- DRD2
- Delta carbonic anhydrase
- Dopamine D1 receptor
- Dopamine receptor
- HTR6
- Histamine H1 receptor
- Muscarinic acetylcholine receptor M2
- Serotonin (5-HT) receptor
- Serotonin receptor 2a and 2c (5HT2A and 5HT2C)
- Sigma non-opioid intracellular receptor 1
- adrenergic Alpha2
- CHEMBL26
- Compound 7
- N-[(1-ethylpyrrolidin-2-yl)methyl]-2-methoxy-5-sulfamoylbenzamide
- SULPIRIDE,(+)
- SULPIRIDE,(-)
- Sulpiride
- Sulpiride, SLP
- Sulpiride-R
- US10172837, Sulpiride
- 3',5'-cyclic phosphodiesterase
- Acetylcholinesterase and butyrylcholinesterase (AChE and BChE)
- Bile salt export pump
- Calcium channel (Type L)
- Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A
- Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B
- Canalicular multispecific organic anion transporter 1
- Canalicular multispecific organic anion transporter 2
- Heart phosphodiesterase
- Homo sapiens phosphodiesterase 2A (PDE2A)
- Multidrug resistance-associated protein 4
- Phosphodiesterase 1
- Phosphodiesterase 11A
- Phosphodiesterase 11A (PDE11A)
- Phosphodiesterase 3
- Phosphodiesterase 3 and 5 (PDE3 and PDE5)
- Phosphodiesterase 4
- Phosphodiesterase 4 and 5 (PDE4 and PDE5)
- Phosphodiesterase 5
- Phosphodiesterase 5A
- Phosphodiesterase 6
- Phosphodiesterase 7
- Phosphodiesterase 8
- Phosphodiesterase 9A
- Phosphodiesterase Type 10 (PDE10A)
- Phosphodiesterase Type 11 (PDE11A)
- Phosphodiesterase Type 2 (PDE2A)
- Phosphodiesterase Type 3 (PDE3B)
- Phosphodiesterase Type 4 (PDE4B)
- Phosphodiesterase Type 4 (PDE4D)
- Phosphodiesterase Type 5 (PDE5A)
- Phosphodiesterase Type 7 (PDE7B)
- Phosphodiesterase Type 9 (PDE9A)
- Potassium voltage-gated channel subfamily H member 2
- Sodium channel protein type 5 subunit alpha
- Voltage-gated potassium channel beta subunit Mink/subunit Kv7.1
- cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A
- cAMP-specific 3',5'-cyclic phosphodiesterase 4B
- cGMP-inhibited 3',5'-cyclic phosphodiesterase B
- cGMP-specific 3',5'-cyclic phosphodiesterase
- (2R,8R)-2-(2H-1,3-benzodioxol-5-yl)-6-methyl-3,6,17-triazatetracyclo[8.7.0.0^{3,8}.0^{11,16}]heptadeca-1(10),11(16),12,14-tetraene-4,7-dione
- (6R,12aR)-6-(1,3-benzodioxol-5-yl)-2-methyl-2,3,6,7,12,12a-hexahydropyrazino[1,2,1,6]pyrido[3,4-b]indole-1,4-dione
- CHEMBL779
- Cialis
- GF 196960
- Tadalafil
- 5-hydroxytryptamine receptor 1A
- 5-hydroxytryptamine receptor 2A
- 5-hydroxytryptamine receptor 2C
- Acetylcholine receptor protein alpha chain/beta chain/delta chain /gamma chain
- Alpha-1A adrenergic receptor
- Alpha-2A adrenergic receptor
- Beta-1 adrenergic receptor
- Beta-2 adrenergic receptor
- Bile salt export pump
- Canalicular multispecific organic anion transporter 1
- Canalicular multispecific organic anion transporter 2
- D(1A) dopamine receptor
- D(2) dopamine receptor
- Gamma-aminobutyric acid receptor subunit alpha-1
- Histamine H1 receptor
- Monoamine transporter
- Multidrug resistance-associated protein 4
- Muscarinic acetylcholine receptor M1
- Muscarinic acetylcholine receptor M2
- Muscarinic acetylcholine receptor M3
- Muscarinic acetylcholine receptor M4
- Muscarinic acetylcholine receptor M5
- Neuronal acetylcholine receptor Alpha-4/Beta-2
- Neuronal acetylcholine receptor protein alpha-3/beta-2 subunit
- Neuronal acetylcholine receptor protein alpha-4/beta-4 subunit
- Neuronal acetylcholine receptor protein alpha-7 subunit
- Neuronal acetylcholine receptor; alpha3/beta4
- Norepinephrine transporter
- Potassium voltage-gated channel subfamily H member 2
- Serotonin receptor 2a and 2c (5HT2A and 5HT2C)
- Sodium-dependent dopamine transporter
- Sodium-dependent noradrenaline transporter
- Sodium-dependent serotonin transporter
- Uridine-5'-diphosphoglucuronosyltransferase 1A1
- Uridine-5'-diphosphoglucuronosyltransferase 1A4
- Uridine-5'-diphosphoglucuronosyltransferase 1A6
- Uridine-5'-diphosphoglucuronosyltransferase 2B10
- Uridine-5'-diphosphoglucuronosyltransferase 2B7
- adrenergic Alpha2
- n-AChR
- 2-(tert-butylamino)-1-(3-chlorophenyl)propan-1-one
- BUPROPION
- BUPROPION HYDROCHLORIDE
- CHEMBL894
- US9944618, Compound ID No. 176
- 3-phosphoinositide dependent protein kinase-1
- ALK tyrosine kinase receptor
- Aurora kinase A/Targeting protein for Xklp2
- Axin-1/Glycogen synthase kinase-3 beta
- Cyclin-Dependent Kinase 4 (CDK4)
- Cyclin-dependent kinase 2
- Ephrin receptor
- Ephrin type-B receptor 4
- Epidermal growth factor receptor
- Fibroblast growth factor receptor 3
- Fibroblast growth factor receptor 4
- Hepatocyte growth factor receptor
- Insulin receptor
- Insulin-like growth factor I receptor
- MAP kinase-activated protein kinase 2
- MAP kinase-interacting serine/threonine-protein kinase 2
- Mast/stem cell growth factor receptor Kit
- Mitogen-activated protein kinase 1
- Mitogen-activated protein kinase 14
- Mitogen-activated protein kinase kinase kinase 8
- Non-receptor tyrosine-protein kinase TYK2
- Platelet-derived growth factor receptor alpha
- Protein kinase C alpha type
- Protein kinase C theta type
- Protein kinase N1
- Protein kinase N2
- Proto-oncogene tyrosine-protein kinase receptor Ret
- Receptor tyrosine-protein kinase erbB-2
- Rho-associated protein kinase 2
- Tyrosine-protein kinase ABL1
- Tyrosine-protein kinase BTK
- Tyrosine-protein kinase JAK1
- Tyrosine-protein kinase JAK2
- Tyrosine-protein kinase JAK3
- Tyrosine-protein kinase Lck
- Tyrosine-protein kinase SYK
- Tyrosine-protein kinase ZAP-70
- Tyrosine-protein kinase receptor UFO
- Vascular endothelial growth factor receptor 2
- cAMP-dependent protein kinase (PKA)
44 IC50
- CHEMBL3786167
- 3-phosphoinositide dependent protein kinase-1
- ALK tyrosine kinase receptor
- Aurora kinase A/Targeting protein for Xklp2
- Axin-1/Glycogen synthase kinase-3 beta
- Cyclin-Dependent Kinase 4 (CDK4)
- Cyclin-dependent kinase 2
- Ephrin receptor
- Ephrin type-B receptor 4
- Epidermal growth factor receptor
- Fibroblast growth factor receptor 3
- Fibroblast growth factor receptor 4
- Hepatocyte growth factor receptor
- Insulin receptor
- Insulin-like growth factor I receptor
- MAP kinase-activated protein kinase 2
- MAP kinase-activated protein kinase 5
- MAP kinase-interacting serine/threonine-protein kinase 2
- Mast/stem cell growth factor receptor Kit
- Mitogen-activated protein kinase 1
- Mitogen-activated protein kinase 14
- Mitogen-activated protein kinase kinase kinase 8
- Non-receptor tyrosine-protein kinase TYK2
- Platelet-derived growth factor receptor alpha
- Potassium voltage-gated channel subfamily H member 2
- Protein kinase C alpha type
- Protein kinase C theta type
- Protein kinase N1
- Protein kinase N2
- Proto-oncogene tyrosine-protein kinase receptor Ret
- Receptor tyrosine-protein kinase erbB-2
- Rho-associated protein kinase 2
- Tyrosine-protein kinase ABL1
- Tyrosine-protein kinase BTK
- Tyrosine-protein kinase JAK1
- Tyrosine-protein kinase JAK2
- Tyrosine-protein kinase JAK3
- Tyrosine-protein kinase Lck
- Tyrosine-protein kinase SYK
- Vascular endothelial growth factor receptor 2
- cAMP-dependent protein kinase (PKA)
44 IC50
- CHEMBL3785500
- ALK tyrosine kinase receptor
- Axin-1/Glycogen synthase kinase-3 beta
- COUP transcription factor 1
- Cyclin-dependent kinase 2
- Epidermal growth factor receptor
- Epidermal growth factor receptor(L858R)
- Epidermal growth factor receptor(L858R, T790M)
- Hepatocyte growth factor receptor
- Insulin receptor
- Insulin-like growth factor I receptor
- Interleukin-1 receptor-associated kinase 4
- Lysyl-tRNA synthetase
- MAP kinase-activated protein kinase 2
- MAP kinase-activated protein kinase 5
- MAP kinase-interacting serine/threonine-protein kinase 1
- MAP kinase-interacting serine/threonine-protein kinase 2
- Macrophage-stimulating protein receptor
- Mast/stem cell growth factor receptor Kit
- Mitogen-activated protein kinase 1
- Mitogen-activated protein kinase 12
- Mitogen-activated protein kinase 14
- Mitogen-activated protein kinase 9
- Non-receptor tyrosine-protein kinase TYK2
- Protein kinase C alpha type
- Protein kinase C theta type
- Protein kinase N1
- Protein kinase N2
- Proto-oncogene tyrosine-protein kinase Src
- RAC-alpha serine/threonine-protein kinase
- Receptor protein-tyrosine kinase erbB-4
- Receptor tyrosine-protein kinase erbB-2
- Rho-associated protein kinase 2
- Serine/threonine-protein kinase PLK1
- Serine/threonine-protein kinase WNK1
- Serine/threonine-protein kinase pim-2
- Tyrosine-protein kinase JAK1
- Tyrosine-protein kinase JAK2
- Tyrosine-protein kinase JAK3
- Vascular endothelial growth factor receptor 2
- [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial
- CHEMBL2178352
- US9096601, 8-26