BDBM100888 US9695132, I-232

SMILES CCC(=O)Nc1cccc(CN2C(=O)C(Cc3cnc(Nc4cccc(NC(=O)C=C)c4)nc23)c2c(Cl)c(OC)cc(OC)c2Cl)c1

InChI Key InChIKey=MSBZHXRISVQJKQ-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 100888   

TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Celgene Car

US Patent
LigandPNGBDBM100888(US9695132, I-232)
Affinity DataIC50: <100nMpH: 7.5Assay Description:Omnia Assay Protocol for Potency Assessment Against FGFR 4 Enzyme. b) [FGFR4-WT]=2.5 nM, [ATP]=250 uM, [Y10-Sox]=10 uM (ATP KMapp 250 uM): A 10x stoc...More data for this Ligand-Target Pair
In DepthDetails US Patent