BDBM104139 US8575145, 16

SMILES C(Oc1cccc2ccc(nc12)-c1nnc2ccccn12)C1CCCNC1

InChI Key InChIKey=FUGPTCJAZZYCRJ-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 104139   

TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM104139(US8575145, 16)
Affinity DataIC50:  1nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-3(Rattus norvegicus (Rat))
Array Biopharma

US Patent
LigandPNGBDBM104139(US8575145, 16)
Affinity DataIC50:  4nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-2(Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM104139(US8575145, 16)
Affinity DataIC50:  169nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails US Patent