BDBM11056 (2S)-1-[(2S)-pyrrolidin-2-ylcarbonyl]pyrrolidine-2-carbonitrile::2-cyanopyrrolidine 10a::CHEMBL381626
SMILES O=C([C@@H]1CCCN1)N1CCC[C@H]1C#N
InChI Key InChIKey=SBKBWYVWRSDAJC-IUCAKERBSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 7 hits for monomerid = 11056
Affinity DataKi: 20nM ΔG°: -10.4kcal/molepH: 7.5 T: 2°CAssay Description:The DPP4 activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 355 nm and mea...More data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:In vitro test for inhibitory activity against human dipeptidyl peptidase IV.More data for this Ligand-Target Pair
Affinity DataIC50: 2.90nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
Affinity DataIC50: 2.90nMAssay Description:Inhibitory concentration against human dipeptidyl-peptidase IVMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90nMAssay Description:Inhibitory concentration against rat dipeptidyl-peptidase IVMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair