BDBM121307 US8722896, (-)-(3R)-1-(Indolin-4-ylmethyl)- N-(9-chloro-2,3,4,5-tetrahydro- 1-benzoxepin-7-ylmethyl)-N- isobutylpyrrolidine-3- carboxamide
SMILES CC(C)CN(Cc1cc(Cl)c2OCCCCc2c1)C(=O)C1CCN(Cc2cccc3NCCc23)C1
InChI Key InChIKey=YBQGGAQYRPBGKV-UHFFFAOYSA-N
Data 3 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 121307
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents of The University of California
US Patent
The Regents of The University of California
US Patent
Affinity DataKi: 0.560nM ΔG°: -13.1kcal/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
TargetProkineticin receptor 1(Cricetulus griseus (Chinese hamster))
The Regents of The University of California
US Patent
The Regents of The University of California
US Patent
Affinity DataKi: 1.56nM ΔG°: -12.5kcal/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
TargetProkineticin receptor 2(Cricetulus griseus (Chinese hamster))
The Regents of The University of California
US Patent
The Regents of The University of California
US Patent
Affinity DataKi: 1.86nM ΔG°: -12.4kcal/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair