BDBM13279 4-{[(3S)-3-[(7-methoxynaphthalene-2-)(methyl)sulfonamido]-2-oxopyrrolidin-1-yl]methyl}thiophene-2-carboximidamide::4-{[(3S)-3-{[(7-methoxynaphthalen-2-yl)sulfonyl](methyl)amino}-2-oxopyrrolidin-1-yl]methyl}thiophene-2-carboximidamide::CHEMBL84638::RPR120844::Sulfonamidopyrrolidinone
SMILES COc1ccc2ccc(cc2c1)S(=O)(=O)N(C)[C@H]1CCN(Cc2csc(c2)C(N)=N)C1=O
InChI Key InChIKey=YQYYTNCSSDRJHZ-IBGZPJMESA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 10 hits for monomerid = 13279
Affinity DataKi: 6.90nM ΔG°: -11.0kcal/molepH: 7.5 T: 2°CAssay Description:The enzyme reactions were initiated by the addition of substrate, and the color developed from the release of p-nitroanilide from each chromogenic su...More data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:In vitro evaluation of inhibitory activity against Coagulation factor X in prothrombinase complexMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Compound was evaluated for the inhibition of human Coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 530nMAssay Description:Inhibitory activity against bovine pancreatic trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Compound was evaluated for the inhibition of thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 2.40E+3nMAssay Description:Compound was evaluated for the inhibition of activated protein C (aPC)More data for this Ligand-Target Pair
Affinity DataKi: 4.40E+3nMAssay Description:Compound was evaluated for the inhibition of plasminMore data for this Ligand-Target Pair
Affinity DataKi: 8.60E+3nMAssay Description:Compound was evaluated for the inhibition of Tissue type plasminogen activator (tissue plasminogen activator)More data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of N-terminus His6-tagged human kallikrein 6 expressed in baculovirus infected insect sf9 cells using Boc-Phe-Ser-Arg-AMC as substrate by ...More data for this Ligand-Target Pair