BDBM146136 US8957068, 171::US8957068, 172
SMILES CC(C)[C@H]1COC(=O)N1c1ccnc(NC(C)c2cccc(F)c2)n1
InChI Key InChIKey=GLVHYTGQNYTKRK-WPZCJLIBSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 146136
Affinity DataIC50: 260nMpH: 7.4 T: 2°CAssay Description:Mutant IDH1 R132H catalytic activity was monitored using the quantitative liquid chromatography/mass spectrometry (LC-MS) detection of 2-HG, a produc...More data for this Ligand-Target Pair
Affinity DataIC50: 6.16E+3nMpH: 7.4 T: 2°CAssay Description:Mutant IDH1 R132H catalytic activity was monitored using the quantitative liquid chromatography/mass spectrometry (LC-MS) detection of 2-HG, a produc...More data for this Ligand-Target Pair