BDBM15471 4-[(1-{[2-oxo-2-(thiophen-3-yl)ethyl]amino}cyclopentyl)methoxy]benzamide::alpha-amino ketone deriv. 12

SMILES NC(=O)c1ccc(OCC2(CCCC2)NCC(=O)c2ccsc2)cc1

InChI Key InChIKey=LMKXIVHWGZZOBT-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 15471   

TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Eli Lilly

LigandPNGBDBM15471(4-[(1-{[2-oxo-2-(thiophen-3-yl)ethyl]amino}cyclope...)
Affinity DataIC50:  5nMpH: 7.5 T: 2°CAssay Description:The DPP activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 355 nm and meas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed