BDBM158333 US9029370, 127
SMILES Fc1cc(NC(=O)c2cnn(c2)-c2cncc(n2)C(F)(F)F)ccc1[C@H]1CNCCO1
InChI Key InChIKey=JWIDABJXMBXRBJ-OAHLLOKOSA-N
Data 2 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 158333
Affinity DataKi: 1.60nM ΔG°: -12.5kcal/molepH: 7.4 T: 2°CAssay Description:HEK-293 cells stably expressing rat TAAR1 were maintained at 37 C and 5% CO2 in DMEM high glucose medium, containing fetal calf serum (10%, heat inac...More data for this Ligand-Target Pair
Affinity DataKi: 7nM ΔG°: -11.6kcal/molepH: 7.4 T: 2°CAssay Description:Membrane Preparation and Radioligand Binding. HEK-293 cells stably expressing mouse TAA 1 were maintained at 37 C and 5% C02 in DMEM high glucose med...More data for this Ligand-Target Pair