BDBM186344 US9163021, 1
SMILES Cc1cc(nn1CC(=O)Nc1cncc(c1)C(=O)c1cn(c2c(F)cncc12)C(C)(C)CO)C(F)(F)F
InChI Key InChIKey=BXEFSUQEJODLSS-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 186344
Affinity DataIC50: 6.32nMAssay Description:Isolated TRK Enzyme assays use the HTRF KinEASE-TK kit (Cisbio Cat#62TK0PEJ) with recombinant His-tagged cytoplasmic domains of each TRK receptor sou...More data for this Ligand-Target Pair