BDBM20370 1-({4-[(1R,5S)-8-azabicyclo[3.2.1]octan-8-yl]-2,5-difluorophenyl}methyl)-3-1H-indazol-4-ylurea::Indazole Analogue, 64

SMILES Fc1cc(N2[C@H]3CC[C@@H]2CCC3)c(F)cc1CNC(=O)Nc1cccc2[nH]ncc12

InChI Key InChIKey=ZNQKOBGZYQOJJS-GASCZTMLSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 20370   

TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM20370(1-({4-[(1R,5S)-8-azabicyclo[3.2.1]octan-8-yl]-2,5-...)
Affinity DataEC50:  21.3nMAssay Description:The functional antagonist activity of compounds at the TRPV1 receptor was determined with a Ca2+ influx assay by measuring the effect on capsaicin (0...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed