BDBM22866 2-(1,3-thiazol-2-yl)ethan-1-amine::2-(2-Thiazolyl)ethanamine::2-(2-aminoethyl)thiazole::2-Thiazolylethylamine::TEA

SMILES NCCc1nccs1

InChI Key InChIKey=TWZOYAWHWDRMEZ-UHFFFAOYSA-N

Data  2 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 22866   

TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
University of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM22866(2-(1,3-thiazol-2-yl)ethan-1-amine | 2-(2-Thiazolyl...)
Affinity DataKi:  8.49E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Vrije Universiteit Amsterdam

LigandPNGBDBM22866(2-(1,3-thiazol-2-yl)ethan-1-amine | 2-(2-Thiazolyl...)
Affinity DataKi: >1.00E+4nM ΔG°: >-7.09kcal/molepH: 7.4 T: 2°CAssay Description:Ligand displacement assays were performed on The SK-N-MC/hH4R cell homogenates. Retained radioactivity was determined by liquid scintillation countin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
University of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM22866(2-(1,3-thiazol-2-yl)ethan-1-amine | 2-(2-Thiazolyl...)
Affinity DataEC50:  6.76E+3nMAssay Description:H1-Histamine receptor agonism on Guinea pig aorta was evaluated (SEM 0.03-0.18)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed