BDBM239877 US9403767, 33
SMILES CNC1(CCC(CN(C)C)(Cc2ccccc2)CC1)c1ccccc1
InChI Key InChIKey=WFDROECRMFIKNH-UHFFFAOYSA-N
Data 2 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 239877
Affinity DataKi: 1.11E+3nM ΔG°: -8.12kcal/moleT: 2°CAssay Description:The affinity to the human μ-opiate receptor was determined in a homogeneous preparation in microtiter plates. For this, dilution series of the res...More data for this Ligand-Target Pair
Affinity DataKi: 3.96E+3nMpH: 7.4Assay Description:The compounds were examined with membranes of recombinant CHO-ORL 1 cells in a receptor binding assay with 3H-nociceptin/orphanin FQ. This test syste...More data for this Ligand-Target Pair