BDBM239927 US9403767, 106
SMILES COc1ccc(CN(C)C2(CCC(CC2)(N(C)C)c2ccccc2)c2ccccc2)cc1
InChI Key InChIKey=ZXNVSIDBFGSRQB-UHFFFAOYSA-N
Data 2 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 239927
Affinity DataKi: 20nMpH: 7.4Assay Description:The compounds were examined with membranes of recombinant CHO-ORL 1 cells in a receptor binding assay with 3H-nociceptin/orphanin FQ. This test syste...More data for this Ligand-Target Pair
Affinity DataKi: 435nM ΔG°: -8.67kcal/moleT: 2°CAssay Description:The affinity to the human μ-opiate receptor was determined in a homogeneous preparation in microtiter plates. For this, dilution series of the res...More data for this Ligand-Target Pair