BDBM261731 1-Fluoro-N-((1S,2S)-2-hydroxycyclohexyl)-4-((6-(1-methyl-1H-pyrazol-4-yl) pyridin-3-yl)methyl)-2-naphthamide::US9708302, 17

SMILES Cn1cc(cn1)-c1ccc(Cc2cc(C(=O)N[C@H]3CCCC[C@@H]3O)c(F)c3ccccc23)cn1

InChI Key InChIKey=BWTRBPPXLSBFLR-DQEYMECFSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 261731   

TargetMuscarinic acetylcholine receptor M1(RAT)
Hoffmann-La Roche

US Patent
LigandPNGBDBM261731(1-Fluoro-N-((1S,2S)-2-hydroxycyclohexyl)-4-((6-(1-...)
Affinity DataEC50:  14nMAssay Description:The assay is designed to select compounds that possess modulator activity at the acetylcholine muscarinic receptor expressed in CHO cells by measurin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM261731(1-Fluoro-N-((1S,2S)-2-hydroxycyclohexyl)-4-((6-(1-...)
Affinity DataEC50:  10nMAssay Description:The assay is designed to select compounds that possess modulator activity at the acetylcholine muscarinic receptor expressed in CHO cells by measurin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent