BDBM268501 N-(6-cyclopropyl-7-(octahydro-1H-4,7-methanoinden-2-yl)methoxy)-[1,2,4]triazolo[4,3-a]pyridin-3-yl)cyclopropanesulfonamide::US9550775, 26::US9550775, 81

SMILES O=S(=O)(Nc1nnc2cc(OCC3CC4C5CCC(C5)C4C3)c(cn12)C1CC1)C1CC1

InChI Key InChIKey=FGGANSUSGJTQLR-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 268501   

TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268501(N-(6-cyclopropyl-7-(octahydro-1H-4,7-methanoinden-...)
Affinity DataIC50:  4nMpH: 7.2Assay Description:The following patch voltage clamp electrophysiology studies were performed on representative compounds of the invention using human embryonic kidney ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268501(N-(6-cyclopropyl-7-(octahydro-1H-4,7-methanoinden-...)
Affinity DataIC50:  3.71nMpH: 7.2Assay Description:The following patch voltage clamp electrophysiology studies were performed on representative compounds of the invention using human embryonic kidney ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent