BDBM268521 N-(7-((4-chloro-3-(trifluoromethyl)phenoxy)methyl)-6-cyclopropyl-[1,2,4]triazolo[4,3-a]pyridin-3-yl)methanesulfonamide::US9550775, 100::US9550775, 45

SMILES CS(=O)(=O)Nc1nnc2cc(COc3ccc(Cl)c(c3)C(F)(F)F)c(cn12)C1CC1

InChI Key InChIKey=PKYOATXJLBGBKJ-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 268521   

TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268521(N-(7-((4-chloro-3-(trifluoromethyl)phenoxy)methyl)...)
Affinity DataIC50:  7nMpH: 7.2Assay Description:The following patch voltage clamp electrophysiology studies were performed on representative compounds of the invention using human embryonic kidney ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268521(N-(7-((4-chloro-3-(trifluoromethyl)phenoxy)methyl)...)
Affinity DataIC50:  7.15nMpH: 7.2Assay Description:The following patch voltage clamp electrophysiology studies were performed on representative compounds of the invention using human embryonic kidney ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent