BDBM269422 (E)-3-(4-((2-(2- ((dimethylamino)methyl) phenyl)-6- hydroxybenzo[b]thiophen- 3-yl)oxy)phenyl)acrylic acid::US10058534, 77
SMILES CN(C)Cc1ccccc1-c1sc2cc(O)ccc2c1Oc1ccc(\C=C\C(O)=O)cc1
InChI Key InChIKey=PPVGAELBQYVJPN-NTEUORMPSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 269422
Affinity DataIC50: 1.40nMpH: 7.4 T: 2°CAssay Description:Plate MCF7 cells at 0.3 million cells/mL (100 l/well) in black, clear-bottom 96-well plates (Greiner, catalog number 655090) in DMEM/F12 media (Gibco...More data for this Ligand-Target Pair
Affinity DataIC50: 44nMpH: 5.1 T: 2°CAssay Description:The ER transcription assay is a reporter assay that is based on the ability of ER to induce transcription from a luciferase reporter gene containing ...More data for this Ligand-Target Pair