BDBM269468 (E)-3-(4-((6-hydroxy-2- (2-(oxetan-3- yl)phenyl)benzo[b] thiophen-3- yl)oxy)phenyl)acrylic acid::US10058534, 123
SMILES OC(=O)\C=C\c1ccc(Oc2c(sc3cc(O)ccc23)-c2ccccc2C2COC2)cc1
InChI Key InChIKey=YUBDDBHWDRWIHA-KPKJPENVSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 269468
Affinity DataIC50: 1.10nMpH: 7.4 T: 2°CAssay Description:Plate MCF7 cells at 0.3 million cells/mL (100 l/well) in black, clear-bottom 96-well plates (Greiner, catalog number 655090) in DMEM/F12 media (Gibco...More data for this Ligand-Target Pair
Affinity DataIC50: 83nMpH: 5.1 T: 2°CAssay Description:The ER transcription assay is a reporter assay that is based on the ability of ER to induce transcription from a luciferase reporter gene containing ...More data for this Ligand-Target Pair