BDBM27174 1H-indol-1-yl tertiary amine, 18::2-{4-[3-({[2-chloro-3-(trifluoromethyl)phenyl]methyl}(2,2-diphenylethyl)amino)propoxy]-1H-indol-1-yl}acetic acid

SMILES OC(=O)Cn1ccc2c(OCCCN(CC(c3ccccc3)c3ccccc3)Cc3cccc(c3Cl)C(F)(F)F)cccc12

InChI Key InChIKey=RHWNXOWPCIQOAH-UHFFFAOYSA-N

Data  2 EC50

PDB links: 1 PDB ID matches this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 27174   

TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Gsk

LigandPNGBDBM27174(1H-indol-1-yl tertiary amine, 18 | 2-{4-[3-({[2-ch...)
Affinity DataEC50:  4nMpH: 7.5 T: 2°CAssay Description:The LXR LiSA measures the ligand-dependent recruitment of a 25 amino acid fragment of the steroid receptor coactivator 1 (SRC1) to the ligand-binding...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Gsk

LigandPNGBDBM27174(1H-indol-1-yl tertiary amine, 18 | 2-{4-[3-({[2-ch...)
Affinity DataEC50:  14nMpH: 7.5 T: 2°CAssay Description:The LXR LiSA measures the ligand-dependent recruitment of a 25 amino acid fragment of the steroid receptor coactivator 1 (SRC1) to the ligand-binding...More data for this Ligand-Target Pair