BDBM274891 N-(6-(7-(Cyclopropanecarbonyl)-2-(4- fluorophenyl)-5,6,7,8-tetrahydroimidazo [1,2- a]pyrazin-3-yl)imidazo[1,2-b]pyridazin-2-yl)-2- fluoroisonicotinamide::US9556179, Compound 469
SMILES Fc1ccc(cc1)-c1nc2CN(CCn2c1-c1ccc2nc(NC(=O)c3ccnc(F)c3)cn2n1)C(=O)C1CC1
InChI Key InChIKey=WBGUAEGUESAJTD-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 274891
Affinity DataIC50: 2.30nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Affinity DataIC50: 12.9nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair