BDBM275792 N-(azetidin-1- ylsulfonyl)-5-chloro- 4-(4-chloro-3- (trifluoromethyl) phenoxy)-2- fluorobenzamide::US10071957, Example 9
SMILES Fc1cc(Oc2ccc(Cl)c(c2)C(F)(F)F)c(Cl)cc1C(=O)NS(=O)(=O)N1CCC1
InChI Key InChIKey=KJDKNKAWFBQABR-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 275792
Affinity DataIC50: 80.7nMpH: 7.4 T: 2°CAssay Description:Preparation of membranes containing recombinantly expressed sodium channels: Frozen recombinant cell pellets were thawed on ice and diluted to 4 time...More data for this Ligand-Target Pair
Affinity DataIC50: 16nMpH: 7.2Assay Description:Patch voltage clamp electrophysiology allows for the direct measurement and quantification of block of voltage-gated sodium channels (NaV's), and...More data for this Ligand-Target Pair