BDBM275811 5-chloro-4-((5-chloro- 6-isobutoxypyridin- 3-yl)oxy)-2-fluoro- N-(pyridin-3-yl- sulfonyl)benzamide::US10071957, Example 28
SMILES CC(C)COc1ncc(Oc2cc(F)c(cc2Cl)C(=O)NS(=O)(=O)c2cccnc2)cc1Cl
InChI Key InChIKey=FWBXSQFYDXIPLL-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 275811
Affinity DataIC50: 703nMpH: 7.4 T: 2°CAssay Description:Preparation of membranes containing recombinantly expressed sodium channels: Frozen recombinant cell pellets were thawed on ice and diluted to 4 time...More data for this Ligand-Target Pair
Affinity DataIC50: 57nMpH: 7.2Assay Description:Patch voltage clamp electrophysiology allows for the direct measurement and quantification of block of voltage-gated sodium channels (NaV's), and...More data for this Ligand-Target Pair