BDBM280408 US10030012, Example 38::ethyl 4-[4-(3- methoxypyridin- 2-yl)piperidin-1- yl]azepane-1- carboxylate
SMILES CCOC(=O)N1CCCC(CC1)N1CCC(CC1)c1ncccc1OC
InChI Key InChIKey=GWGLXRCCVIVRSY-UHFFFAOYSA-N
Data 4 EC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 280408
Affinity DataEC50: 30nMAssay Description:The functional activity of compounds at the M4 and M2 receptors was determined by measuring changes in the level of intracellular calcium ions caused...More data for this Ligand-Target Pair
Affinity DataEC50: 11nMAssay Description:Agonist activity at human Muscarinic acetylcholine receptor M4 expressed in HEK cells co-expressing Glosensor construct assessed as decrease in isopr...More data for this Ligand-Target Pair
Affinity DataEC50: 2.52E+3nMAssay Description:Agonist activity at human Muscarinic acetylcholine receptor M2 expressed in HEK cells co-expressing Glosensor construct assessed as decrease in isopr...More data for this Ligand-Target Pair