BDBM284994 N-[4-methyl-3-(2-methyl-1-oxoisoquinolin- 4-yl)phenyl]methanesulfonamide::US10023592, Example 39
SMILES Cc1ccc(NS(C)(=O)=O)cc1-c1cn(C)c(=O)c2ccccc12
InChI Key InChIKey=RYGKANGIHXJREX-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 284994
Affinity DataIC50: <500nMpH: 7.3Assay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BRD4 was cloned, expr...More data for this Ligand-Target Pair