BDBM285027 N-[3-[2-methyl-6-(6-methylpyridin-3-yl)-1- oxoisoquinolin-4-yl]phenyl]ethanesulfonamide::US10023592, Example 72::US10941160, Example 72
SMILES CCS(=O)(=O)Nc1cccc(c1)-c1cn(C)c(=O)c2ccc(cc12)-c1ccc(C)nc1
InChI Key InChIKey=ILUWENTYMZHYSD-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 285027
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BRD4 was cloned, expr...More data for this Ligand-Target Pair
Affinity DataIC50: <500nMpH: 7.3Assay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BRD4 was cloned, expr...More data for this Ligand-Target Pair