BDBM285283 5-[3-[(2,6-dimethylphenyl)methoxy]-5- methylsulfonylphenyl]-1,3- dimethylpyridin-2-one::BDBM486127::US10023592, Example 331
SMILES Cc1cccc(C)c1COc1cc(cc(c1)S(C)(=O)=O)-c1cc(C)c(=O)n(C)c1
InChI Key InChIKey=IOKGUKBEUPWMBT-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 285283
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BRD4 was cloned, expr...More data for this Ligand-Target Pair
Affinity DataIC50: <500nMpH: 7.3Assay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BRD4 was cloned, expr...More data for this Ligand-Target Pair