BDBM285292 5-(3-but-2-ynoxy-5-methylsulfonylphenyl)-1,3- dimethylpyridin-2-one::BDBM486136::US10023592, Example 340
SMILES CC#CCOc1cc(cc(c1)S(C)(=O)=O)-c1cc(C)c(=O)n(C)c1
InChI Key InChIKey=SDCQIFQDDJKRKX-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 285292
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BRD4 was cloned, expr...More data for this Ligand-Target Pair
Affinity DataIC50: <500nMpH: 7.3Assay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BRD4 was cloned, expr...More data for this Ligand-Target Pair