BDBM292043 3-(1H-Indazol-5-yl)-2-(pyridin-2-yl)-5-(trifluoromethyl)-2H-pyrazolo[4,3-b]pyridine;::US10100045, Example 14

SMILES FC(F)(F)c1ccc2nn(c(-c3ccc4[nH]ncc4c3)c2n1)-c1ccccn1

InChI Key InChIKey=GUKFIBJBKYTUKV-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 292043   

TargetVoltage-dependent calcium channel gamma-2 subunit(Homo sapiens (Human))
Janssen Pharmaceutica

US Patent
LigandPNGBDBM292043(3-(1H-Indazol-5-yl)-2-(pyridin-2-yl)-5-(trifluorom...)
Affinity DataIC50:  126nMpH: 7.4Assay Description:Cell expressing the GRIA1o-CACNG8 fusion construct were grown in a monolayer in 96- or 384-well microtiter plates. They were washed with assay buffer...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent