BDBM293563 US10106527, Compound 273::US10544128, Compound 273::US10604514, Compound 76::US11548872, Compound 273::US20230286945, Compound 273::US9951048, Compound 273
SMILES Cn1cncc1-c1ccc2cnc(NC(=O)c3ccnc(c3)N3CCOCC3)cc2c1
InChI Key InChIKey=ZABAYWAGMFKGHJ-UHFFFAOYSA-N
Data 12 EC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 293563
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Samumed
US Patent
Samumed
US Patent
Affinity DataEC50: 1.10nMT: 2°CAssay Description:Briefly, recombinant DYRK1A kinase, ATP and Ser/Thr peptide 18 were prepared in 1× Kinase buffer to final concentrations of 0.19 μg/mL, 30 μ...More data for this Ligand-Target Pair
Affinity DataEC50: 2.90E+3nMT: 2°CAssay Description:Briefly, recombinant GSK3β kinase, ATP and Ser/Thr peptide 09 are prepared in 1× Kinase buffer to final concentrations of 0.04 μg/mL, 46 ...More data for this Ligand-Target Pair