BDBM297530 US10118902, Example 32::US10584103, Example 32::[4-[4-(2-azetidin-1-yl-phenyl)- piperidin-1-yl]-2-(1-methyl- cyclopropyl)-quinazolin-6-yl]- methyl-(2-morpholin-4-yl-ethyl)- amine

SMILES CN(CCN1CCOCC1)c1ccc2nc(nc(N3CCC(CC3)c3ccccc3N3CCC3)c2c1)C1(C)CC1

InChI Key InChIKey=LJOJMWATPLOZIY-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 297530   

TargetNeurotensin receptor type 1(Homo sapiens (Human))
Sanford Burnham Prebys Medical Discovery Institute

US Patent
LigandPNGBDBM297530(US10118902, Example 32 | US10584103, Example 32 | ...)
Affinity DataEC50: >1.00E+4nMAssay Description:NTSR1 (NTR1) CHO cells are plated in 20 μL of assay media containing Ham's F12 supplemented with 10% fetal bovine serum and 0.4 mg/mL G418 a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Sanford Burnham Prebys Medical Discovery Institute

US Patent
LigandPNGBDBM297530(US10118902, Example 32 | US10584103, Example 32 | ...)
Affinity DataEC50: >1.00E+4nMAssay Description:NTSR1 (NTR1) CHO cells are plated in 20 uL of assay media containing Ham's F12 supplemented with 10% fetal bovine serum and 0.4 mg/mL G418 at a c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent