BDBM300803 3-[4-[[3-(2- Methylphenyl)benzo[b]thiophen- 5-yl]methoxy]phenyl] propanoic acid::US10131648, Compound 1::US10195178, Compound 1::US9790198, Compound 1

SMILES Cc1ccccc1-c1csc2ccc(COc3ccc(CCC(O)=O)cc3)cc12

InChI Key InChIKey=CUNNWYSORXWPNQ-UHFFFAOYSA-N

Data  3 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 300803   

TargetFree fatty acid receptor 1(Homo sapiens (Human))
Janssen Pharmaceutica

US Patent
LigandPNGBDBM300803(3-[4-[[3-(2- Methylphenyl)benzo[b]thiophen- 5-yl]m...)
Affinity DataEC50:  7nMAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Janssen Pharmaceutica

US Patent
LigandPNGBDBM300803(3-[4-[[3-(2- Methylphenyl)benzo[b]thiophen- 5-yl]m...)
Affinity DataEC50:  7nMAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Janssen Pharmaceutica

US Patent
LigandPNGBDBM300803(3-[4-[[3-(2- Methylphenyl)benzo[b]thiophen- 5-yl]m...)
Affinity DataEC50:  7nMAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent