BDBM329063 4-(6-(3-chloro-4- methylphenoxy)-5-cyano-3- pyridinyl)-3-methoxy-N- (methylsulfonyl)benzamide::4-(6-(3-chloro-4-methylphenoxy)-5-cyano-3-pyridinyl)-3-methoxy-N-(methylsulfonyl)benzamide::US9663508, Example 549::US9663508, Example 829

SMILES COc1cc(ccc1-c1cnc(Oc2ccc(C)c(Cl)c2)c(c1)C#N)C(=O)NS(C)(=O)=O

InChI Key InChIKey=AZNREZPQQMFMKF-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 329063   

TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Amgen

US Patent
LigandPNGBDBM329063(4-(6-(3-chloro-4- methylphenoxy)-5-cyano-3- pyridi...)
Affinity DataIC50:  50.5nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Amgen

US Patent
LigandPNGBDBM329063(4-(6-(3-chloro-4- methylphenoxy)-5-cyano-3- pyridi...)
Affinity DataIC50:  50.5nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent