BDBM329077 4-(5-Chloro-6-(2,4-Dichloro-6-Methylphenoxy)-Pyridin-3-yl)-3-Methoxy-N-(Methylsulfonyl)Benzamide::4-(5-chloro-6-(2,4-dichloro-6-methylphenoxy)-3-pyridinyl)-3-methoxy-N-(methylsulfonyl)benzamide::US9663508, Example 578

SMILES COc1cc(ccc1-c1cnc(Oc2c(C)cc(Cl)cc2Cl)c(Cl)c1)C(=O)NS(C)(=O)=O

InChI Key InChIKey=AWDNJCGXGVQTBS-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 329077   

TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Amgen

US Patent
LigandPNGBDBM329077(4-(5-Chloro-6-(2,4-Dichloro-6-Methylphenoxy)-Pyrid...)
Affinity DataIC50:  29.6nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent