BDBM329097 5-chloro-4-(5-chloro-6-(2,4-dichloro-6-methylphenoxy)-3-::5-chloro-4-(5-chloro-6-(2,4-dichloro-6-methylphenoxy)-3-pyridinyl)-2-fluoro-N-(methylsulfonyl)benzamide::US9663508, Example 598

SMILES Cc1cc(Cl)cc(Cl)c1Oc1ncc(cc1Cl)-c1cc(F)c(cc1Cl)C(=O)NS(C)(=O)=O

InChI Key InChIKey=RBBAYENCPUYUIC-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 329097   

TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Amgen

US Patent
LigandPNGBDBM329097(5-chloro-4-(5-chloro-6-(2,4-dichloro-6-methylpheno...)
Affinity DataIC50:  18.4nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent