BDBM329192 4-(5-cyano-6-(3,6-dichloro-2-methylphenoxy)-3-pyridinyl)-3-methoxy-N-(methylsulfonyl)benzamide::US9663508, Example 694

SMILES COc1cc(ccc1-c1cnc(Oc2c(Cl)ccc(Cl)c2C)c(c1)C#N)C(=O)NS(C)(=O)=O

InChI Key InChIKey=LSFXTMIQOHAEEG-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 329192   

TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Amgen

US Patent
LigandPNGBDBM329192(4-(5-cyano-6-(3,6-dichloro-2-methylphenoxy)-3-pyri...)
Affinity DataIC50:  17.2nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent