BDBM34159 indenylsulfonamide, 47+48::isomeric mixture (70% 5-indenyl, 30% 6-indenyl)

SMILES CC1=Cc2cc(NS(=O)(=O)c3c(Cl)nc4sccn34)ccc2C1

InChI Key InChIKey=LZIANNQBBHNPFV-UHFFFAOYSA-N

Data  1 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 34159   

Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universitat De Barcelona

LigandPNGBDBM34159(indenylsulfonamide, 47+48 | isomeric mixture (70% ...)
Affinity DataKi:  43nM ΔG°:  -10.4kcal/mole IC50:  3.00E+3nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed using membranes from HEK-293 transfected with human 5-HT6 receptor. In these membranes the receptor concent...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed