BDBM349139 4-[2-(Cyclopropanecarbonyl- amino)-[1,2,4]triazolo[1,5- a]pyridin-5-yl]-N-(1,1-dioxo- tetrahydrothiophen-3-yl)-N- methyl-benzamide::US10206907, Compound 273
SMILES CN(C1CCS(=O)(=O)C1)C(=O)c1ccc(cc1)-c1cccc2nc(NC(=O)C3CC3)nn12
InChI Key InChIKey=MVZJDAIADOAREM-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 349139
Affinity DataIC50: <100nMAssay Description:Recombinant human JAK1 catalytic domain (amino acids 850-1154; catalog number 08-144) was purchased from Carna Biosciences. 10 ng of JAK1 was incubat...More data for this Ligand-Target Pair
Affinity DataIC50: <100nMAssay Description:Recombinant human JAK2 catalytic domain (amino acids 808-1132; catalog number PV4210) was purchased from Invitrogen. 0.025 mU of JAK2 was incubated w...More data for this Ligand-Target Pair