BDBM375228 3-bromo-6-(pyridin-3-yl)-5-(pyridin-4-yl)pyridin-2-amine::US10253017, Example 22
SMILES Nc1cc(Br)c(-c2ccncc2)c(n1)-c1cccnc1
InChI Key InChIKey=IPWUMLNQSJDQEN-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 375228
Affinity DataKi: 46.1nMAssay Description:The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...More data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...More data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:The experiment of binding to MT3 sites was carried out on hamster brain membranes using [125I]2-iodomelatonin as radioligand in accordance with the p...More data for this Ligand-Target Pair