BDBM375229 3-chloro-5-(3-fluoropyridin-4-yl)-6-(pyridin-3-yl)pyridin-2-amine::US10253017, Example 23
SMILES Nc1cc(Cl)c(-c2ccnc(F)c2)c(n1)-c1cccnc1
InChI Key InChIKey=JNYHGOGFLOVUNA-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 375229
Affinity DataKi: 23.9nMAssay Description:The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...More data for this Ligand-Target Pair
Affinity DataKi: 4.80E+3nMAssay Description:The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...More data for this Ligand-Target Pair
Affinity DataIC50: 98nMAssay Description:The experiment of binding to MT3 sites was carried out on hamster brain membranes using [125I]2-iodomelatonin as radioligand in accordance with the p...More data for this Ligand-Target Pair