BDBM387354 N-[2-(6-methylpyridin-2-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]-1H-indazol-5-amine::US10292985, Example 36
SMILES Cc1cccc(n1)-c1nc(Nc2ccc3[nH]ncc3c2)c2cccn2n1
InChI Key InChIKey=FFIOTQBLWQNPEJ-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 387354
Affinity DataIC50: 1.5nMAssay Description:Assays are conducted in 1536-well plates and 2 mL reactions are prepared from addition of HIS-TGFβR1 T204D or HIS-TGFβR2 WT, anti-HIS detec...More data for this Ligand-Target Pair