BDBM392391 3,4-dimethyl-N-(3-methyl-1H- pyrazolo[3,4-b]pyridin-5-yl)-1H- pyrazole-5-carboxamide::US10301280, Compound P-2040
SMILES Cc1n[nH]c(C(=O)Nc2cnc3[nH]nc(C)c3c2)c1C
InChI Key InChIKey=ANERYXRMFWJMKO-UHFFFAOYSA-N
Data 2 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 392391
Affinity DataKi: <1.00E+3nMAssay Description:The c-kit mutant D816V (or kinase domain thereof) is an active kinase in AlphaScreen. IC50 values are determined with respect to inhibition of c-Kit ...More data for this Ligand-Target Pair
Affinity DataKi: 1.05E+5nMAssay Description:Assays for biochemical cell-based activity of c-kit kinase are known in the art, for example, as described in U.S. Pat. Nos. 7,498,342 and 7,846,941,...More data for this Ligand-Target Pair