BDBM392409 3-methyl-N-(2-morpholino-1H- pyrrolo[2,3-b]pyridin-5-yl)-1H- pyrazole-5-carboxamide::US10301280, Compound P-2058

SMILES Cc1cc([nH]n1)C(=O)Nc1cnc2[nH]c(cc2c1)N1CCOCC1

InChI Key InChIKey=FFJCKOMDADUPIX-UHFFFAOYSA-N

Data  2 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 392409   

TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Plexxikon

US Patent
LigandPNGBDBM392409(3-methyl-N-(2-morpholino-1H- pyrrolo[2,3-b]pyridin...)
Affinity DataKi: <1.00E+3nMAssay Description:The c-kit mutant D816V (or kinase domain thereof) is an active kinase in AlphaScreen. IC50 values are determined with respect to inhibition of c-Kit ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMast/stem cell growth factor receptor Kit [D816V](Homo sapiens (Human))
Plexxikon

US Patent
LigandPNGBDBM392409(3-methyl-N-(2-morpholino-1H- pyrrolo[2,3-b]pyridin...)
Affinity DataKi:  1.05E+5nMAssay Description:Assays for biochemical cell-based activity of c-kit kinase are known in the art, for example, as described in U.S. Pat. Nos. 7,498,342 and 7,846,941,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent