BDBM392488 3-[5-[(3,4-dimethyl-1H-pyrazole-5- carbonyl)amino]-1H-pyrrolo[2,3- b]pyridin-2-yl]pyridine-4- carboxamide::US10301280, Compound P-2272
SMILES Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2cnccc2C(N)=O)c1C
InChI Key InChIKey=RZABNWWGCMXMAO-UHFFFAOYSA-N
Data 2 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 392488
Affinity DataKi: <1.00E+3nMAssay Description:The c-kit mutant D816V (or kinase domain thereof) is an active kinase in AlphaScreen. IC50 values are determined with respect to inhibition of c-Kit ...More data for this Ligand-Target Pair
Affinity DataKi: 1.05E+5nMAssay Description:Assays for biochemical cell-based activity of c-kit kinase are known in the art, for example, as described in U.S. Pat. Nos. 7,498,342 and 7,846,941,...More data for this Ligand-Target Pair